平安! 发表于 2011-11-9 19:57
: n. Y# o. j( {Pazopanib (100 mg/kg/day free base equivalent)
9 T/ k5 Y" r; R; S* L 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。2 d- d8 W3 r7 M9 T
搜索了一下,原料一大堆。% B2 L9 F) |% a
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对不起!100mg/kg是用于移植瘤的,我弄错了。$ `8 W6 Q- ?# e6 v
5 q& b/ T5 V/ d( e以下是正版说明书的推荐用量。) X1 o9 d: z1 b* y/ q4 u
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--------------------- DOSAGE AND ADMINISTRATION ----------------1 `2 Z+ m |" {) v- P, V
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 3 }" J: |, h+ p. l0 v. A
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) . b- Y U' ^* A$ f6 X
---------------------DOSAGE FORMS AND STRENGTHS --------------
! b3 J t* Q1 _, F200 mg tablets. (3) ; o4 \' c# {, F7 v, H, M8 m7 u, U
-------------------------------CONTRAINDICATIONS------------------------ |